G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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Items 161-170 of 247

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  1. Description:

    5-HT4 receptor agonist. Also 5-HT3 antagonist.

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $141
    Qty:
    Pack:
    50mg
    Price:
    $565
    Qty:
  2. Description:

    Potent, selective mGluR5 antagonist / mGluR4 positive allosteric modulator

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $118
    Qty:
    Pack:
    50mg
    Price:
    $439
    Qty:
  3. Description:

    Selective P2Y1 antagonist. Inhibits platelet aggregation.

    Purity:

    >98%

    Pack:
    5mg
    Price:
    $113
    Qty:
    Pack:
    10mg
    Price:
    $209
    Qty:
    Pack:
    50mg
    Price:
    $911
    Qty:
  4. MRS 2578 (HB1966)

    Description:

    Potent, selective P2Y6 receptor antagonist

    Purity:

    >95%

    Pack:
    10mg
    Price:
    $134
    Qty:
  5. MS 245 oxalate (HB1782)

    Description:

    5-HT6 antagonist

    Purity:

    >99%

    Pack:
    50mg
    Price:
    $617
    Qty:
  6. Pack:
    10mg
    Price:
    $128
    Qty:
    Pack:
    50mg
    Price:
    $483
    Qty:
    Pack:
    10mM (add 1ml water)
    Price:
    $50
    Qty:
  7. Pack:
    200μg
    Price:
    $123
    Free trial
    Qty:
    Pack:
    500μg
    Price:
    $260
    Qty:
    Pack:
    1mg
    Price:
    $499
    Qty:
  8. Description:

    Invertebrate neurotransmitter. Chemogenetic DmOctβ1 receptor activator.

    Purity:

    >99%

    Pack:
    1g
    Price:
    $31
    Qty:
    Pack:
    5g
    Price:
    $90
    Qty:
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