G protein coupled receptors

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G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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Items 1-10 of 240

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  1. 2  Reviews
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    Description:

    Neurotoxin, widely used to produce the 6-OHDA Parkinson’s disease model

    Purity:

    >98%

    Pack:
    50mg
    Price:
    $55
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    Pack:
    250mg
    Price:
    $104
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    Pack:
    1g
    Price:
    $349
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  2. A 83-01 (HB3218)

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    Description:

    Selective TGF-βRI (ALK5), ALK4 and ALK7 inhibitor. Maintains human hiPSC self renewal, 3D growth matrix component and promotes long-term organoid growth. Aids fibroblast to NSC/cardiomyocyte reprogramming.

    Purity:

    >98%

    Pack:
    5mg
    Price:
    $80
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    Pack:
    25mg
    Price:
    $270
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  3. Description:

    Potent dopamine D4 receptor partial agonist

    Purity:

    >99%

    Pack:
    50mg
    Price:
    $568
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  4. Pack:
    10mg
    Price:
    $243
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    Pack:
    50mg
    Price:
    $917
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  5. AM251 (HB2776)

    3  Reviews
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    Description:

    Potent, selective CB1 receptor antagonist / inverse agonist

    Purity:

    >98%

    Pack:
    1mg
    Price:
    $56
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    Pack:
    10mg
    Price:
    $124
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    Pack:
    50mg
    Price:
    $476
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  6. Pack:
    10mg
    Price:
    $152
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    Pack:
    50mg
    Price:
    $626
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  7. L-AP4 (HB0370)

    3  Reviews
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    Description:

    L-AP4 is a selective group III mGluR agonist which inhibits synaptic transmission.

    Purity:

    >99%

    Pack:
    5mg
    Price:
    $74
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    Pack:
    10mg
    Price:
    $143
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    Pack:
    25mg
    Price:
    $298
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    Pack:
    50mg
    Price:
    $592
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