G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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  1. Description:

    Potent dopamine D4 receptor partial agonist

    Purity:

    >99%

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    50mg
    Price:
    $644
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    100mg
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    $240
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    10mg
    Price:
    $87
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    50mg
    Price:
    $386
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  4. L-AP4 (HB0370)

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    Description:

    L-AP4 is a selective group III mGluR agonist which inhibits synaptic transmission.

    Purity:

    >99%

    Pack:
    5mg
    Price:
    $102
    Free trial
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    10mg
    Price:
    $197
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    25mg
    Price:
    $411
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    Price:
    $816
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  5. Pack:
    10mg
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    $69
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    $284
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    Pack:
    25mM (add 1ml water)
    Price:
    $100
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  6. Description:

    5-HT1A partial agonist

    Pack:
    10mg
    Price:
    $85
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    50mg
    Price:
    $308
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  7. BRL 54443 (HB1664)

    Description:

    Potent 5-ht1E/1F receptor agonist

    Pack:
    10mg
    Price:
    $150
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    50mg
    Price:
    $516
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