Target

Highly potent, selective, competitive dipeptidyl-peptidase 4 inhibitor

K_v7 channel blocker

Potent MGMT inhibitor

Mitochondrial hexokinase inhibitor

Potent, selective µ-opioid receptor agonist

Potent and selective HIV-1 protease inhibitor

Selective, non-peptide AT₁ antagonist

Selective I₂-imidazoline receptor ligand

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, covalent Affinity-Based Probe (AfBP). Clickable antagonist for the A₂AR.