Target

Potent, selective K_ir1.1 channel blocker

Non-selective K⁺ channel blocker

Potent, selective, use-dependent Na⁺ channel blocker. Citrate free.

Potent, selective, use-dependent Na⁺ channel blocker. Citrate Salt.

Potent, selective K_Ca3.1 channel blocker

TRPV2 channel inhibitor. Potent mast cell stabilizer.

Novel, potent, subtype-selective TRPV3 inhibitor

Potent, selective, reversible T-type calcium channel blocker

Selective TRPA1 activator

L-type Ca²⁺ channel blocker