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Tertiapin LQ

(HB1107)
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Product overview

Name Tertiapin LQ
Purity >95%
Description Potent, selective Kir1.1 channel blocker
Biological Data Solubility & Handling Chemical Data Related Areas Calculators Technical guides (1) Reviews References (1) Frequently bought together
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Images

Tertiapin LQ product vial image | Hello Bio
Tertiapin LQ product vial image | Hello Bio

Tertiapin LQ product vial image | Hello Bio

Tertiapin LQ product vial image | Hello Bio

Biological Data

Biological description Tertiapin-Q derivative. Potent and selective Kir1.1 channel blocker. Selective for Kir1.1 over Kir3.1/3.2 and Kir3.1/3.4 (Kd values are 1.1, 274 and 361 nM respectively).

Solubility & Handling

Storage instructions -20°C
Solubility overview Soluble in acetonitrile (2mg/ml)
Important This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

Calculators

Molarity

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More Info

Dilution

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Chemical Data

Purity >95%
Molecular Weight 2428.03
Molecular Formula C106H179N33O24S4
PubChem identifier 90488935
SMILES [H]N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3=CNC4=C3C=CC=C4)NC2=O)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CC(N)=O)NC1=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC
InChiKey WUMIWMIQOSXVPZ-ZPWFPUPGSA-N

References for Tertiapin LQ

References are publications that support the biological activity of the product

  • Engineered specific and high-affinity inhibitor for a subtype of inward-rectifier K+ channels.

    Ramu Y et al (2008) Proc Natl Acad Sci U S A 105(31) : 10774-8.
    Read more (PubMedID: 18669667)

1 Item

Grouped product items
Order: HB1107
Pack PriceQty
1mg
$161
Potent, selective Kir1.1 channel blocker
Shipping Info

Standard: $35

Hazardous: $35

Shipped on ice: $35

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