Target

K_v7 channel blocker

Potent, non-selective K_v1.3 channel blocker

Non-competitive NMDA receptor antagonist

Potent, selective α7 nicotinic receptor antagonist

Potent, reversible T- / L-type Ca²⁺ channel blocker

K_ir6 channel activator

Potent, selective, non-competitive NMDA receptor antagonist

Less active enantiomer of (+)-MK 801. NMDA receptor antagonist.

Selective K_v7.2 / K_v7.4 channel activator

Selective K_2P2.1 (TREK-1) and K_2P10.1 (TREK-2) activator