GluN2C

Potent, selective, competitive glycine site NMDA receptor antagonist

Competitive, selective EAAT2 inhibitor

Selective H₂ receptor agonist

Cell-permeable, redox cycling quinone. Induces ROS generation.

Selective, competitive AMPA / kainate receptor antagonist

Selective, competitive AMPA / kainate receptor antagonist. Sodium salt.

Selective ERβ estrogen receptor agonist

Effective agonist for muscarinic-based DREADDs in vitro and in vivo. Non-CNO chemogenetic actuator. Brain penetrant. Water soluble.

Effective agonist for muscarinic-based DREADDs in vitro and in vivo. Non-CNO chemogenetic actuator. Brain penetrant.

Novel selective estrogen-related receptor ERRβ and ERRγ agonist