Novel selective estrogen-related receptor ERRβ and ERRγ agonist. Shows no effect on ERRα or ERRα/β. Inhibits proliferation of prostate cancer cells. Blood brain barrier permeable.
Solubility & Handling
Storage instructions
+4°C
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.
K2P2.1 (TREK-1) modulator. Used with ML336 as part of the CATKLAMP chemogenetic strategy. Selectively and irreversibly activates TREK-1CG* but not wild-type K2P2.1 (TREK-1)