GluN2

PD-1/PD-L1 interaction inhibitor

Potent, highly selective iNOS inhibitor

IP₃ receptor and store-operated channels (SOC) channel antagonist

Aurora B and C kinase inhibitor

Potent, cell-permeable calmodulin (CaM) antagonist

Potent, selective Na_v1.8 channel inhibitor

Selective TGF-βRI (ALK5), ALK4 and ALK7 inhibitor. Maintains human hiPSC self renewal, 3D growth matrix component and promotes long-term organoid growth. Aids fibroblast to NSC/cardiomyocyte reprogramming.

Potent, selective TRPA1 channel blocker

Selective cPLA₂ inhibitor

Selective Hsp90 inhibitor. Also protects neuroprogenitor cells against apoptosis.