c-Src

Potent CaM kinase II inhibitor

Potent, selective PKA inhibitor

Potent, selective PKG inhibitor

Potent, selective mTOR inhibitor

Potent, selective, irreversible proteasome inhibitor

Acyl-CoA cholesterol acyltransferase (ACAT) inhibitor

Potent, non-selective tyrosine kinase inhibitor

Reversible trypsin-like and cysteine proteases inhibitor

Highly potent, selective, competitive dipeptidyl-peptidase 4 inhibitor

Potent MGMT inhibitor