Inflammasome

Mitochondrial hexokinase inhibitor

Potent, selective µ-opioid receptor agonist

Potent and selective HIV-1 protease inhibitor

Selective, non-peptide AT₁ antagonist

Selective I₂-imidazoline receptor ligand

Chemiluminescent luciferase substrate

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, covalent Affinity-Based Probe (AfBP). Clickable antagonist for the A₂AR.

Novel, intracellular covalent chemokine CCR2 negative allosteric modulator (NAM). Binds irreversibly.

Novel, potent, selective A₃AR covalent antagonist