TLR7

Potent mGlu₅ positive allosteric modulator

Potent, selective ATP-competitive p38 MAPK inhibitor

Potent, selective p38α MAPK inhibitor

Calmodulin (CaM) antagonist

Potent 5-HT_1A receptor antagonist. D₄ receptor agonist.

Selective IKKα and IKKβ kinase activity inhibitor. NF-κB inhibitor.

Non-selective JAK3 inhibitor and potent EGFR inhibitor. Induces neural progenitor cell differentiation.

Lipodepsipeptide with antibacterial, antifungal and antimicrobial activity

Potent tankyrase inhibitor. Wnt signaling inhibitor.

Potent, selective N-WASP inhibitor