5-HT2

Jumonji histone demethylase inhibitor

Downstream Hedgehog signaling pathway inhibitor. Alcohol dehydrogenase 7 inhibitor.

Potent, selective H₄ receptor silent antagonist

Potent, selective, non-competitive mGlu₁ antagonist

Potent, selective BET bromodomain inhibitor. Cell permeable.

Potent, reversible p38α MAPK inhibitor

Non-selective protein kinase inhibitor

Potent PKC and casein kinase II inhibitor

PKC inhibitor

Prototypic, selective kainate receptor agonist. Potent excitant and neurotoxin.