DNA methyltransferase (DNMT)

Selective antagonist for GluN2D subunit containing NMDA receptors

Highly potent, selective GluN2C/2D NMDAR antagonist

Potent, selective GluK1 subunit selective kainate receptor antagonist

Potent, selective GluK1 / GluK3 subunit selective kainate receptor antagonist

UCPH-101 is a potent, selective, non-competitive EAAT1 inhibitor

Selective EAAT1 inhibitor

Topoisomerase II inhibitor

Potent, selective G9a HMTase inhibitor

Potent, selective G9a / GLP HMTase inhibitor

Selective 5-HT_1A agonist. α₁-adrenoceptor antagonist