DNA methyltransferase (DNMT)

Potent, selective protein phosphatase 1 / 2A inhibitor

Serine protease inhibitor. Inhibits TMPRSS2 and partially blocks SARS-Cov2 entry in vitro.

Potent, selective PP2A inhibitor

ACE and LTA₄ hydrolase inhibitor

NO scavenger

Anti-oxidant, anti-inflammatory compound with many actions. Topoisomerase II inhibitor.

Potent and specific PKC inhibitor

Selective CDK1 inhibitor

Potent histone methyltransferase SUV39H1 inhibitor

Monoamine oxidase (MAO) inhibitor