HMG-CoA synthase

Potent, selective, non-competitive mGlu₁ antagonist

Potent, selective BET bromodomain inhibitor. Cell permeable.

Potent, reversible p38α MAPK inhibitor

Non-selective protein kinase inhibitor

Potent PKC and casein kinase II inhibitor

PKC inhibitor

Selective, reverse mode Na⁺ / Ca²⁺ exchange inhibitor

Atypical voltage-gated sodium channel blocker

Potent endothelin receptor antagonist

Potent CDK inhibitor. Also GSK-3 inhibitor. Generates iPSCs.