Secretase

Non-selective group I/II mGluR antagonist

Non-selective group I and II mGluR antagonist. Water soluble sodium salt.

Water soluble, non-selective group I and II mGluR antagonist

Selective mGlu₈ receptor antagonist

Potent and selective 5-HT_2A receptor antagonist

Free fatty acid 1 (FFA₁) receptor agonist

Inhibits α-MSH release inhibitors. Also increase dopamine levels.

Non-competitive NMDA receptor antagonist

Selective H₁ receptor inverse agonist

5-HT₁/5-HT₂ antagonist. Shows affinity for 5-HT₆ and 5-HT₇.