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G-protein receptor kinases (GRKs) help terminate GPCR signaling through receptor desensitization and downregulation and also modulate signaling via phosphorylation-independent functions. GRKs affect various physiological processes. Researchers can save up to 50% on GRK modulators from Hello Bio - they are around half the price of other suppliers.
10Z-Hymenialdisine (HB1264)
Description:Pan kinase inhibitor. Potently inhibits MEK1, Cdk1, Cdk2, Cdk3 and Cdk5 and GSK-3β.
Purity:>97%
Ibrutinib (HB4204)
Description:Potent, selective Bruton's tyrosine kinase (BTK) inhibitor.
Purity:>98%
Imatinib mesylate (HB1943)
Description:Tyrosine kinase inhibitor that targets BCR‑ABL, c‑KIT, and PDGFR kinases
Purity:>98%