Target

Mouse excitatory neuropeptide at orexin OX₁/OX₂ receptors

Reproductive hormone. Neuropeptide.

PAR₄ antagonist. Inhibits platelet aggregation.

5-HT_2A and D₂ antagonist. Antipsychotic.

TLR2/6 activator. Induces potent NF-κB activation and cytokine production.

TLR1/TLR2 agonist and potent NF-κB activator. Induces cytokine production.

Potent, selective serotonin reuptake inhibitor. Selective GRK2 inhibitor.

Potent, selective M₄ receptor antagonist. Promotes erythroid progenitors expansion.

FGFR1/ FGFR3 inhibitor. Inhibits oligodendrocyte progenitor proliferation and differentiation.

Effective agonist for muscarinic-based DREADDs in vitro and in vivo. Non-CNO chemogenetic actuator