p38 MAPK

Standard D₂-like dopamine receptor antagonist

Actin filament inhibitor. Disrupts actin cytoskeleton.

Potent, p-38 MAP kinase inhibitor. Wnt/β-catenin signaling inhibitor.

Selective, non-competitive AMPA / kainate receptor antagonist

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

Selective D₁-D₂ heteromer antagonist

Cx43 hemichannel blocker. Active in vivo.

GluK6-PSD-95 interaction inhibitor

Competitive EAAT blocker. Inhibits glutamate uptake.