Hedgehog signaling

Potent, selective H₄ receptor silent antagonist

Potent, selective, non-competitive mGlu₁ antagonist

Potent, selective BET bromodomain inhibitor. Cell permeable.

Potent, reversible p38α MAPK inhibitor

Non-selective protein kinase inhibitor

Potent PKC and casein kinase II inhibitor

PKC inhibitor

Prototypic, selective kainate receptor agonist. Potent excitant and neurotoxin.

Protein synthesis inhibitor. Broad spectrum antibiotic.

Potently induces chondrogenesis in MSCs