Immunology & Inflammation

Potent, selective, non-competitive mGlu₁ antagonist

Potent, reversible p38α MAPK inhibitor

Potent endothelin receptor antagonist

Selective 5-HT₂ receptor antagonist

Potent, selective mTOR inhibitor

Immediate precursor of dopamine

Potent, non-selective tyrosine kinase inhibitor

Potent and selective ACKR3 (CXCR7) agonist. Potentiates opioid peptide activity.

Potent, selective µ-opioid receptor agonist

Selective, non-peptide AT₁ antagonist