ROCK (Rho-kinase)

Potent, p-38 MAP kinase inhibitor. Wnt/β-catenin signaling inhibitor.

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

AT₁ antagonist and PPARγ partial agonist

DNA-methylating antitumor agent

Antibacterial phytotoxin

Antibiotic with antibacterial and anticancer activity

Selective PAR₁ activating peptide

Potent, non-competitive SERCA inhibitor

Phytotoxin. Plant cell necrosis inducer.