Mineralocorticoid

Peripheral dopamine D₂-like receptor antagonist

Potent AChE inhibitor

Water soluble L-DOPA derivative

Potent, selective AMPK inhibitor. Promotes neural hPSCs differentiation and promotes cardiomyocyte differentiation in mESCs.

Antibiotic. DNA topisomerase II inhibitor. Apoptosis inducer.

Broad-spectrum antibiotic. Used in inducible Tet-on/ Tet-off gene expression systems for gene editing.

Potent, selective A₁ receptor inverse agonist

Selective ERβ estrogen receptor agonist

Highly potent PARP-1 inhibitor

Effective agonist for muscarinic-based DREADDs in vitro and in vivo. Non-CNO chemogenetic actuator. Brain penetrant. Water soluble.