Mineralocorticoid

Selective D₁-D₂ heteromer antagonist

Competitive EAAT blocker. Inhibits glutamate uptake.

Potent and selective orexin OX₂ antagonist

5-HT₄ partial agonist

AT₁ antagonist and PPARγ partial agonist

Potent inhibitor of vesicular monoamine transport; depletes 5-HT stores

Selective PAR₁ activating peptide

Amino acid analog of Glutamine. Promotes hESC self-renewal.

Adenosine receptor antagonist

Selective GAT-1 GABA uptake inhibitor