DREADD

Filters

Designer receptors exclusively activated by designer drugs (DREADDs) are genetically engineered GPCRs that are activated by physiologically inert synthetic small molecules (designer drugs) but not their endogenous ligand. Read our DREADDs mini-review or for practical advice on using these ligands in the lab see Stability of Water-Soluble DREADD Ligands in Solution: A Technical Review and Clozapine N-Oxide (freebase) - a technical review on stability, solubility and use in the lab).

Items 411-420 of 747

Set Descending Direction
  1. Description:

    Potent, selective α7 nicotinic receptor antagonist

    Purity:

    >95%

    Pack:
    5mg
    Price:
    $70
    Qty:
    Pack:
    25mg
    Price:
    $259
    Qty:
  2. MG132 (HB4135)

    Description:

    Potent, cell-permeable proteasome inhibitor. Calpain inhibitor. Apoptosis inducer.

    Purity:

    >95%

    Pack:
    5mg
    Price:
    $103
    Free trial
    Qty:
    Pack:
    25mg
    Price:
    $300
    Qty:
  3. MHY 1485 (HB7154)

    Description:

    mTOR activator and autophagy inhibitor. Cell-permeable.

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $58
    Qty:
    Pack:
    50mg
    Price:
    $182
    Qty:
  4. Pack:
    5mg
    Price:
    $113
    Qty:
    Pack:
    10mg
    Price:
    $201
    Qty:
    Pack:
    25mg
    Price:
    $474
    Qty:
  5. Mifepristone (HB2783)

    Description:

    Potent glucocorticoid and progesterone receptor antagonist. Also used for gene editing as a mifepristone inducible Cas9 and Cpf1 CRISPR effector.

    Purity:

    >99%

    Pack:
    100mg
    Price:
    $85
    Qty:
  6. Description:

    5-HT and norepinephrine re-uptake inhibitor (SNRI)

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $122
    Qty:
    Pack:
    50mg
    Price:
    $432
    Qty:
  7. Pack:
    25mg
    Price:
    $87
    Qty:
    Pack:
    50mg
    Price:
    $132
    Qty:
    Pack:
    100mg
    Price:
    $197
    Qty:
    Pack:
    500mg
    Price:
    $783
    Qty:
  8. Description:

    Highly selective, pan-Akt inhibitor. Autophagy and apoptosis inducer. Orally bioavailable.

    Purity:

    >98%

    Pack:
    5mg
    Price:
    Qty:
    Pack:
    10mg
    Price:
    $77
    Qty:
    Pack:
    50mg
    Price:
    $325
    Qty:
    Pack:
    10mM solution (in 1mL DMSO)
    Price:
    $125
    Qty:
  9. Description:

    Selective leukotriene LTD4 receptor antagonist. Potent MRP1 inhibitor.

    Purity:

    >97%

    Pack:
    25mg
    Price:
    $276
    Qty:
  10. Pack:
    10mg
    Price:
    $59
    Qty:
    Pack:
    50mg
    Price:
    $260
    Qty:
    Pack:
    20mM (add 1ml water)
    Price:
    $74
    Qty:
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