Toll-like receptor

K_2P2.1 (TREK-1) modulator. Selectively and irreversibly activates TREK-1^CG* but not wild-type K_2P2.1 (TREK-1)

Selective mGlu₅ positive allosteric modulator

Selective M₁ receptor agonist

Potent STING ligand

Prototypic, selective A_2A receptor agonist

Antibiotic with antibacterial, antifungal and cytotoxic activity. Selectively induces apoptosis of CLL cells.

Macrolide antibiotic with antimicrobial and antibacterial activity

Antimalarial. Apoptosis and autophagy inhibitor.

Selective mGluR₅ agonist. Water soluble sodium salt.

Selective mGlu₅ agonist