Toll-like receptor

IκB kinase inhibitor. NF-κB inhibitor.

Selective PPARγ agonist

Selective mGlu₄ agonist

GluN2C / GluN2D subunit selective NMDA receptor positive allosteric modulator

Mitochondrial permeability transition pore (MPTP) activator

Antibiotic. Protein synthesis inhibitor

Prototypic, atypical antipsychotic, binds to both serotonin and dopamine receptors

Water soluble prototypic, atypical antipsychotic. Binds to both serotonin and dopamine receptors.

Prototypical DREADD activator. Clozapine metabolite.

Dihydrochloride salt of CNO - the prototypical DREADD activator