Receptors & Transporters

PKC inhibitor

Glycoside with various biological actions

Selective, competitive CaM-KK inhibitor

Potent, p-38 MAP kinase inhibitor. Wnt/β-catenin signaling inhibitor.

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

Cx43 hemichannel blocker. Active in vivo.

Abundant free amino acid found in the brain.

AT₁ antagonist and PPARγ partial agonist

Potent, non-competitive SERCA inhibitor