GluN2

Ceramide-activated protein phosphatase (CAPP) activator

TRPV1 channel agonist

K_2P2.1 (TREK-1) modulator. Selectively and irreversibly activates TREK-1^CG* but not wild-type K_2P2.1 (TREK-1)

Selective mGlu₅ positive allosteric modulator

Selective M₁ receptor agonist

Potent STING ligand

Prototypic, selective A_2A receptor agonist

Selective NMDA receptor antagonist

Antimalarial. Apoptosis and autophagy inhibitor.

Selective mGluR₅ agonist. Water soluble sodium salt.