DNA methyltransferase (DNMT)

GluK6-PSD-95 interaction inhibitor

Competitive EAAT blocker. Inhibits glutamate uptake.

Selective class I HDAC inhibitor

Potent, selective Na_v1.7 inhibitor

Potent, non-competitive GluN2A subunit selective NMDA receptor antagonist

Potent and selective orexin OX₂ antagonist

5-HT₄ partial agonist

Acyl-CoA cholesterol acyltransferase 1 and 2 inhibitor

Potent, specific, irreversible acetylcholinesterase (AChE) inhibitor.

Potent inward rectifier K⁺ channel blocker