TLR7

PI3K/AKT/mTOR signaling inhibitor. Antitumour activity.

Potent, selective guanylyl cyclase inhibitor

Potent, non-competitive protein phosphatase inhibitor

Water soluble, potent protein phosphatase 1 and 2A inhibitor

5-HT_2A and D₂ antagonist. Potent DREADD agonist. Atypical antipsychotic.

LPA1 and LPA2 agonist. Inhibits differentiation of neural stem cells (NSCs) into neurons.

PLA₂ inhibitor

Inhibitor of mitochondrial function

Farnesyltransferase (FTase) inhibitor

Potent, selective P-type / Q-type Ca²⁺ channel blocker