PI3K/Akt/mTOR

Fluorogenic tri-peptide substrate. Useful for measuring trypsin-like 20S proteasome peptidase activity.

Highly potent, selective, cell permeable proteasome inhibitor. More potent than MG-132.

Potent, reversible and cell permeable proteasome inhibitor

Reversible and cell permeable proteasome inhibitor

Potent, selective A_2A receptor antagonist

Potent, selective, ATP-competitive Aurora kinase B inhibitor

Potent 5-HT_1B/1D/1F agonist

Potent, selective Na⁺ / H⁺ exchanger-1 inhibitor

Non-selective Na⁺ / Ca²⁺ channel blocker

5-HT_2A and dopamine D₂ receptor antagonist. Atypical antipsychotic.