Mineralocorticoid

Adenosine receptor antagonist

Selective GAT-1 GABA uptake inhibitor

Selective 5-HT uptake enhancer

Potent, selective PPARγ agonist. Inhibits hematopoietic cell line growth.

Novel NMDAR pan-PAM

NMDAR pan-PAM that potentiates all GluN2 subunits. Enhances LTD and decreases LTP. 

NMDAR PAM which potentiates GluN2A and GluN2B with minimal effects on 2C and 2D.

UCPH-101 is a potent, selective, non-competitive EAAT1 inhibitor

Selective EAAT1 inhibitor

Selective TRPA1 activator