Mineralocorticoid

Potent GABA_B receptor agonist

Selective glucagon receptor antagonist. Non-peptidic anti-diabetic agent

PAR₂ peptide agonist

Selective TRPML3 channel activator

Regulatory neuropeptide

Activates the hFFA2-DREADD

Selective mGlu₃ agonist, peptide neurotransmitter

nNOS inhibitor / PTPN₂ activator

Selective D₂-like receptor antagonist. 5-HT_2A antagonist.

Mineralocorticoid and androgen receptor antagonist