Aurora kinase

Selective D₂-like receptor antagonist. 5-HT_2A antagonist.

Mineralocorticoid and androgen receptor antagonist

Potent,selective, cell permeable yeast NAD+-dependent HDAC Sir2p inhibitor

Potent, selective ROCK inhibitor

Selective, competitive GABA_A receptor antagonist

Selective STAT3 inhibitor

Potent, non-specific protein kinase inhibitor. Apoptosis inducer.

PKC inhibitor

Phytosterol with anticancer and many other biological actions. Farnesoid X receptor antagonist.

Selective, competitive CaM-KK inhibitor