Non-selective

Selective class I HDAC inhibitor

Potent, selective Na_v1.7 inhibitor

Potent, non-competitive GluN2A subunit selective NMDA receptor antagonist

Potent and selective orexin OX₂ antagonist

5-HT₄ partial agonist

Acyl-CoA cholesterol acyltransferase 1 and 2 inhibitor

Potent, specific, irreversible acetylcholinesterase (AChE) inhibitor.

Potent inward rectifier K⁺ channel blocker

Potent, selective K_ir1.1 channel blocker

Potent inhibitor of vesicular monoamine transport; depletes 5-HT stores