ROCK (Rho-kinase)

Pancreatic, gastric and carboxylester lipase inhibitor

Selective Na⁺ / K⁺ ATPase inhibitor. Shows antiviral activity.

Reproductive hormone. Neuropeptide.

PAR₄ antagonist. Inhibits platelet aggregation.

Procaspase-activating compound

5-HT_2A and D₂ antagonist. Antipsychotic.

Rasfarnesyltransferase inhibitor

TLR2/6 activator. Induces potent NF-κB activation and cytokine production.

TLR1/TLR2 agonist and potent NF-κB activator. Induces cytokine production.

Potent, selective serotonin reuptake inhibitor. Selective GRK2 inhibitor.