Agonists & activators
An agonist or activator, is a drug or chemical that binds to and activates a protein, such as receptor or enzyme. Full agonists have high efficacy, eliciting a full response whilst occupying a small proportion of receptors. Partial agonists have a lower efficacy and cannot produce a maximal response, even if occupying a high proportion of receptors. Inverse agonists can bind to the same receptor binding-site as an agonist, but elicit an opposite effect. Researchers can save up to 50% on activators, agonists, partial agonists and inverse agonists from Hello Bio - they are up to half the price of other suppliers.
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Fluorescent M3 muscarinic receptor antagonist
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Fluorescent GABAB receptor antagonist
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Fluorescent 5-HT1A receptor antagonist
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Fluorescent 5-HT2A receptor antagonist
LUF7487 (HB9585)
Description:Novel, covalent Affinity-Based Probe (AfBP). Clickable antagonist for the A2AR.
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Novel, intracellular covalent chemokine CCR2 negative allosteric modulator (NAM). Binds irreversibly.