GluN2

Phytotoxin. Derivative of the HDAC inhibitor chlamydocin.

5-HT antagonist. Also partial agonist at adrenergic and dopaminergic receptors.

Partial α-adrenergic agonist, partial D₂ agonist and 5-HT antagonist

Competitive, selective EAAT2 inhibitor

PKC inhibitor

Selective H₂ receptor agonist

Shows no COX-2 inhibitory function. Analog of celecoxib.

Reversibly stimulates SERCA Ca²⁺-ATPase. V-ATPase inhibitor.

Selective ALK2 inhibitor. Promotes iPSC neurogenesis.

Cell-permeable, redox cycling quinone. Induces ROS generation.