HMG-CoA synthase

Potent aldose reductase inhibitor

Selective PP1R15A inhibitor

Phosphodiesterase 4 (PDE4) inhibitor with various biological actions

Potent, selective 5-HT re-uptake inhibitor (SSRI)

Bacterial DNA gyrase inhibitor

Na⁺ / Ca⁺ channel blocker

Potent, competitive NOS inhibitor

Potent, selective D₁-like receptor antagonist

Potent, selective, competitive GAT-1 GABA uptake inhibitor

Selective glucagon receptor antagonist. Non-peptidic anti-diabetic agent