Hedgehog signaling

Novel, intracellular covalent chemokine CCR2 negative allosteric modulator (NAM). Binds irreversibly.

Novel, potent, selective A₃AR covalent antagonist

The first covalent hA₁AR partial agonist. Binds Irreversibly.

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Novel, clickable Adenosine hA₃AR Affinity-Based Probe (AfBP).

Novel Selective A_2B covalent ligand. Binds irreversibly.

Antiparasitic compound. Also shows cytotoxic activity.

Chemiluminiscent compound

Potent, highly selective mGlu_1a antagonist. Water soluble.

High affinity, selective 5-HT_2B receptor antagonist