TLR7

Potent, selective PKA inhibitor

Potent, selective mTOR inhibitor

Endogenous ionotropic glutamate / nicotinic antagonist.

Na²⁺ / K⁺ / Ca²⁺ channel inhibitor. Anticonvulsant.

Actin polymerization inhibitor

Potent and selective ACKR3 (CXCR7) agonist. Potentiates opioid peptide activity.

Inhibits protein synthesis in gram-positive bacteria. Antibiotic.

Peptide fragment of LL-37 (human)

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, covalent Affinity-Based Probe (AfBP). Clickable antagonist for the A₂AR.