GluN2

Selective M₁ receptor agonist

Antimalarial. Apoptosis and autophagy inhibitor.

Selective mGlu₄ agonist

Mitochondrial permeability transition pore (MPTP) activator

Water soluble prototypic, atypical antipsychotic. Binds to both serotonin and dopamine receptors.

Dihydrochloride salt of CNO - the prototypical DREADD activator

Potent, selective, competitive NMDA receptor antagonist

Potent NMDA receptor antagonist

mGlu_1α / mGlu_5a agonist

Potent, selective and metabolically stable hM3Dq and hM4Di muscarinic DREADD actuator.