Mineralocorticoid

Major metabolite of GLP-1 (7-36)

Dopamine receptor antagonist with partial D₂-like selectivity

Synthetic estrogen receptor ligand. Widely used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Synthetic estrogen receptor ligand. Widely used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor ligand. For inducible genome manipulation (e.g. Cre-LoxP (CreER)/ TRAP/ CRISPR-Cas9).

Selective TRPC6 channel activator and neurotransmitter re-uptake inhibitor

Non-selective endogenous glycine receptor agonist 

Potent TRPM8 channel agonist

Potent muscarinic acetylcholine receptor superagonist. Also binds the hM3R-miniG_q DREADD receptor.

Piezo1 channel activator