Dopamine receptor antagonist with partial D2-like receptor selectivity (Ki values are 0.53, 2.7, 2.3, 27 and 48 nM at D2, D3, D4, D1 and D5 receptors respectively).
Shows variety of biological actions. Active in vivo.
Recently investigated as part of COVID-19 compound repurposing.
Solubility & Handling
Solubility overview
Soluble in DMSO (20 mM with warming), and in ethanol (10 mM with warming)
Storage instructions
Room temperature
Storage of solutions
Prepare and use solutions on the same day if possible. Store solutions at -20°C for up to one month if storage is required. Equilibrate to RT and ensure the solution is precipitate free before use.
Shipping Conditions
Stable for ambient temperature shipping. Follow storage instructions on receipt.
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.