Receptors & Transporters

Novel, potent, selective A₃AR covalent antagonist

Potent, highly selective mGlu_1a antagonist. Water soluble.

5-HT_1D-preferring receptor antagonist

Potent, highly selective mGlu_1a antagonist

Non-selective group I and II mGluR antagonist

Non-selective group I/II mGluR antagonist

Non-selective group I and II mGluR antagonist. Water soluble sodium salt.

Water soluble, non-selective group I and II mGluR antagonist

Potent and selective 5-HT_2A receptor antagonist

Non-selective 5-HT₂ receptor antagonist. Shows activity at other receptors.