Histone demethylase

Potent, selective, non-competitive NMDA receptor antagonist

Novel caged, fast-equilibrating glutamate receptor antagonist. Suitable for use as a synaptic probe.

5-HT₄ receptor agonist. Also 5-HT₃ antagonist.

Potent, selective mGluR₅ antagonist / mGluR₄ positive allosteric modulator

Selective ERα estrogen receptor antagonist

Selective P2Y₁ antagonist. Inhibits platelet aggregation.

Potent, selective P2Y₆ receptor antagonist

Potent, highly selective, non-competitive mGluR₅ antagonist

Selective GluA2- lacking, Ca²⁺ permeable AMPA / kainate receptor antagonist

Potent, selective, competitive AMPA receptor antagonist