PI3K/Akt/mTOR

Estrogen receptor ligand. For inducible genome manipulation (e.g. Cre-LoxP (CreER)/ TRAP/ CRISPR-Cas9).

Selective TRPC6 channel activator and neurotransmitter re-uptake inhibitor

Non-selective endogenous glycine receptor agonist 

Potent, reversible, selective K_Ca channel inhibitor

Potent, selective Bruton's tyrosine kinase (BTK) inhibitor.

Potent, selective Na_v1.3 / Na_v1.1 channel inhibitor

Potent, selective cAMP PDE inhibitor

Potent TRPM8 channel agonist

Potent muscarinic acetylcholine receptor superagonist. Also binds the hM3R-miniG_q DREADD receptor.

Piezo1 channel activator